BREAKING
PROSETTA WINS ARPA-H "DASH TO ACCELERATE HEALTH OUTCOMES" PAV-615 SHOWS EFFICACY IN C9orf72 ALS/FTD MODEL NEW PAPER IN CELL REPORTS MEDICINE - OXIDIZED MIF AS ALZHEIMER'S TARGET $31M SERIES D BACKED BY TAKEDA & ALGER MANAGEMENT NCI COLLABORATION ON "ONE DRUG FOR ALL CANCERS" 24-PERSON SF BIOTECH RUNNING SIX THERAPEUTIC PROGRAMS PROSETTA WINS ARPA-H "DASH TO ACCELERATE HEALTH OUTCOMES" PAV-615 SHOWS EFFICACY IN C9orf72 ALS/FTD MODEL NEW PAPER IN CELL REPORTS MEDICINE - OXIDIZED MIF AS ALZHEIMER'S TARGET $31M SERIES D BACKED BY TAKEDA & ALGER MANAGEMENT NCI COLLABORATION ON "ONE DRUG FOR ALL CANCERS" 24-PERSON SF BIOTECH RUNNING SIX THERAPEUTIC PROGRAMS
Profile - Biotech - San Francisco

Prosetta Biosciences

A 24-person biotech in SoMa is screening for drugs the rest of the industry can't see. Their tool: a tube of liquid that builds proteins from scratch. Their target: the unruly committees of molecules behind cancer, ALS, Alzheimer's, and the next pandemic.

Prosetta Biosciences logo
SHELF MARK PBS-01 // The logo of a quiet lab on 5th Street. Inside, the test tubes are doing the talking.
Dispatch

The screen that finds drugs nobody else is looking for.

Walk past 670 5th Street on most days and you'd never guess what's happening inside. No glass atrium. No oat-milk cafeteria. Just a small team, a few benches, and a robot that brews proteins in a test tube and watches what tiny molecules do to them.

Most pharmaceutical screens look for one molecule, locking onto one other molecule. Prosetta looks for chaperoned committees - the multi-protein complexes a cell quietly stitches together when it builds a virus, a tumor, a tangled neuron. The company calls these targets "assemblies." Its founder spent two decades at UCSF arguing they were druggable. Now there's a pipeline trying to prove it.

It's not glamorous biotech. It's stubborn biotech.

By The Numbers

A small lab with a wide aperture.

$66M
Total raised
$31M
Series D, 2015
$35M+
Government contracts
23 yrs
Operating since 2003

Pipeline focus (relative investment, est.)

Oncology
92%
ALS / FTD
80%
Antivirals
68%
Alzheimer's
60%
Biodefense
45%
The Platform

Cell-free protein synthesis, weaponized.

In a normal pharma screen, you pick a target - a single protein - and throw a library of small molecules at it. The catch: many of biology's most important machines are not single proteins. They're assemblies. Twenty proteins that latch together briefly, do something terrible, then dissolve.

Prosetta's platform, CFPSA, builds those assemblies on demand in a tube. A small molecule that nudges the assembly off its course becomes a candidate drug. The platform produces hits that look invisible to conventional screens - not because they're rare, but because nobody's been watching for them.

1. Brew the assembly

A cell-free system synthesizes the target multi-protein complex from RNA. No living cells. No noise.

2. Screen the disruptors

Libraries of small molecules are perturbed against the assembly to find ones that shift its structure or kinetics.

3. Translate to disease

Hits move into cell, animal, and (eventually) clinical models across viruses, cancer, and neurodegeneration.

"A new approach to drug discovery." - the entire homepage, refreshingly stingy with adjectives.
The Pipeline

Six programs. One mechanism.

Most biotechs are companies built around a disease. Prosetta is built around a mechanism. The result: a pipeline that crosses oncology, neurology, virology, and biodefense without flinching.

CNS

PAV-615

An assembly modulator with preclinical efficacy in C9orf72-associated ALS/FTD mouse models and human iPSC-derived motor neurons. Presented at Target ALS 2025.

ONCOLOGY

"One Drug for All Cancers"

The proposal that won the ARPA-H Dash competition in 2023 and led to an NCI collaboration. Small-molecule modulators showing pan-cancer selective cytotoxicity.

ALZHEIMER'S

Oxidized MIF

Cell Reports Medicine, Dec 2025: oxidized MIF relays external risk factors to tau pathology - a fresh angle on a notoriously crowded target landscape.

The Founder

Vishwanath Lingappa, MD, PhD.

He joined the UCSF faculty in 1982 as a physician-scientist and ran an NIH-funded basic research lab for 22+ years. He didn't leave academia in a hurry. He left because he thought the assemblies he kept watching in his lab were medicine waiting to be made.

Today he is Founder, Chief Technology Officer, and Co-CEO. Many founders pivot. He kept the question.

"Our therapeutics work with the body's natural regulatory systems to restore molecular homeostasis."
The Notebook

23 years, in dispatches.

2003

Prosetta is founded by UCSF and UW academics around the cell-free protein synthesis idea.

2010s

Antiviral lead series active against influenza, HIV, HCV emerge from the platform.

Dec 2015

$31M Series D private placement closes - Alger Management and Takeda Pharmaceutical Company among investors.

2023

ARPA-H Dash to Accelerate Health Outcomes win for the "One Drug for All Cancers" oncology program; collaboration with the National Cancer Institute follows.

Dec 2024

Publications on pan-cancer assembly modulator cytotoxicity and on ALS-relevant assembly modulators.

Apr 2025

Clinical Proteomics paper: an ALS assembly modulator signature in peripheral blood mononuclear cells. Diagnostics in the wings.

May 2025

PAV-615 ALS/FTD data presented at Target ALS annual meeting.

Dec 2025

Twin publications: oxidized MIF in Alzheimer's (Cell Reports Medicine) and PAV-615 preclinical evaluation (Cells).

For The Reader

What can you actually do with this?

If you're a scientist

Read the Cell Reports Medicine and Clinical Proteomics papers. The CFPSA approach is open to interrogation.

If you're a patient advocate

Watch the ALS/FTD and Alzheimer's programs. PAV-615 and the MIF work are early but moving.

If you're an investor

Series D was 2015. The next round, if it comes, will be a tell on platform vs. asset framing.

If you're a partner

The NCI collaboration is the template. Prosetta runs on alliances and non-dilutive contracts.

Allies

Who Prosetta runs with.

The cap table is small. The collaborator list, less so. Government agencies, academic labs, and a couple of big pharma names have spent real time inside the platform.

  • + National Cancer Institute - oncology collaboration
  • + Takeda Pharmaceutical Company - strategic investor
  • + Alger Management - lead Series D investor
  • + Target ALS - research community
  • + MTEC - Medical Technology Enterprise Consortium
  • + BARDA / NIH / DoD - non-dilutive contracts
Culture

A lab that thinks like a lab.

Prosetta is the rare biotech where "we publish" is a culture statement, not a press line. The team is small, the meetings are short, the papers are real. Half scrappy startup, half university group that grew teeth.

Six programs. Twenty-four people. One thesis - held longer than most marriages.
Watch & Read

Talks, demos, and deeper cuts.

Coda

Back to 670 5th Street.

The lab on 5th Street still doesn't look like much from the sidewalk. The robot still brews proteins on demand. The team still publishes more than it tweets.

What's different now is that the screen behind the door has produced an Alzheimer's mechanism paper, an ALS candidate moving through models, a pan-cancer program with a federal partner, and a quiet argument: that the next era of medicine will come from drugs that influence committees of proteins, not lone ones. Prosetta has been making that argument for 23 years. The literature finally seems ready to listen.

If they're right, the test tubes on 5th Street will eventually become drugs. If they're wrong, they will at least have demanded that drug discovery look harder at what cells are actually doing - which is, in the end, the only job basic biology ever signed up for.

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Contact & Channels

Where to find Prosetta.